Abstracts

Scientific Abstracts:























COMMON COLD
(Page 3)


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Table of Contents

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book [The effect of astragalus polysaccharides (APS) on cell mediated immunity (CMI) in burned mice]
book Immunomodulating Chinese herbal medicines.
book [The effect of vitamin A and Astragalus on the splenic T lymphocyte-CFU of burned mice]
book Nutritional antioxidants and the modulation of inflammation: theory and practice.
book Evaluation of zinc complexes on the replication of rhinovirus 2 in vitro.
book Zinc gluconate and the common cold: a controlled clinical study.
book Prophylaxis and treatment of rhinovirus colds with zinc gluconate lozenges.
book Reduction in duration of common colds by zinc gluconate lozenges in a double-blind study.
book Antivirals for the chemoprophylaxis and treatment of influenza.
book Utilization of pulse oximetry for the study of the inhibitory effects of antiviral agents on influenza virus in mice.
book Further studies with short duration ribavirin aerosol for the treatment of influenza virus infection in mice and respiratory syncytial virus infection in cotton rats.
book High dose-short duration ribavirin aerosol treatment--a review.
book Viral pneumonia.
book Aerosol and intraperitoneal administration of ribavirin and ribavirin triacetate: pharmacokinetics and protection of mice against intracerebral infection with influenza A/WSN virus.
book Antiviral drug therapy.
book Molecular mechanisms of action of ribavirin.
book New acquisitions in the chemotherapy of viral infections.
book Comparison of oral and aerosol ribavirin regimens in the high risk elderly.
book Comparative activities of several nucleoside analogs against influenza A, B, and C viruses in vitro.
book Antiviral drugs for common respiratory diseases. What's here, what's to come.
book Oral ribavirin treatment of influenza A and B.
book Clinical review of ribavirin.
book Clinical use of antiviral drugs.
book Protection of mice from lethal influenza virus infection with high dose-short duration ribavirin aerosol.
book Ribavirin: a clinical overview.
book Effect of ribavirin triphosphate on primer generation and elongation during influenza virus transcription in vitro.
book Ribavirin
book [Immunomodulating activity of ethanol-water extracts of the roots of Echinacea gloriosa L., Echinacea angustifolia DC. and Rudbeckia speciosa Wenderoth tested on the immune system in C57BL6 inbred mice]
book Application of purified polysaccharides from cell cultures of the plant Echinacea purpurea to mice mediates protection against systemic infections with Listeria monocytogenes and Candida albicans.
book Macrophage activation by the polysaccharide arabinogalactan isolated from plant cell cultures of Echinacea purpurea.
book Macrophage activation and induction of macrophage cytotoxicity by purified polysaccharide fractions from the plant Echinacea purpurea.
book Combined antiviral and antimediator treatment of rhinovirus colds.
book [Common cold: diagnostic steps? Antibiotics?]
book Alpha 2-interferon for the common cold.
book Managing viral upper respiratory infections.
book Immunological barriers in the nose and paranasal sinuses.
book Interferon for the treatment of infections.
book Effect of Astragalus membranaceus on electrophysiological activities of acute experimental coxsackie B-3 viral myocarditis in mice
book Efficacy and safety of the standardized ginseng extract G 115 for potentiating vaccination against common cold and/or influenza syndrome
book An emerging green pharmacy: Modern plant medicines and health
book Immunity in myocardiac hypertrophy rat and effect of total saponins of panax ginseng in vivo and in vitro
book Treatment of experimental coxsackie B-3 viral myocarditis with astragalus membranaceus in mice
book Effect of Astragalus membranaceus injecta on coxsackie b-2 virus infected rat beating heart cell culture
book Sambucol(tm) inhibited several strains of influenza virus and reduced symptoms during an outbreak of Influenza B Panama
book The effect of Sambucol(tm) on HIV infection in vitro


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[The effect of astragalus polysaccharides (APS) on cell mediated immunity (CMI) in burned mice]

Liang H, Zhang Y, Geng B
Research Institute of Surgery, Third Military Medical College, Chongqing.
Chung Hua Cheng Hsing Shao Shang Wai Ko Tsa Chih 1994 Mar;10(2):138-41

In this paper, the changes in CMI in mice were determined after burn injury, and the effects of APS on CMI of burned mice were investigated in vivo. The results showed that on day 6 postburn, spleen index and thymus index were reduced, T lymphocyte transformation and interleukin 2 (IL-2) production were suppressed. Furthermore, the serum and macrophages from burned mice showed significant suppressive activity upon T lymphocyte transformation in vitro, and suppressive index (SI) of suppressor T cell (Ts) was greater than that of normal controls. Intraperitoneal administration of APS (250mg/kg daily, from day 0 to 5 could restore spleen index and thymus index of burned mice, reverse the suppression of T lymphocyte transformation and IL-2 production, reduce remarkably the suppressive activity of serum, macrophages and Ts. It is suggested that (1) burn injury-induced suppression of CMI may be related to the augmented suppressive activity of serum, macrophages and Ts; (2) administration of APS may restore the impaired CMI after burn injury by reducing the suppressive activity of postburn serum, macrophages and Ts.



Immunomodulating Chinese herbal medicines.

Li XY
Shanghai Institute of Materia Medica, Chinese Academy of Sciences.
Mem Inst Oswaldo Cruz (Brazil) 1991, 86 Suppl 2 p159-64

Traditional Chinese medicine always pays close attention to the strengthening of the patient's general resistance against illness, there are many Chinese herbs used for thousands of years are considered as tonics. Animal experiments and modern clinical trails have shown that quite a number herbs are immunologically active, and most of the tonics are excellent immunomodulating agents, such as polysaccharides or saponins isolated from Astragalus mongholicus, Acanthopanax senticosus and Panax notoginseng, which stimulated macrophages, promoted antibody formation, activated complement and increased T lymphocyte proliferation. Moreover, some of them were proved to be anti-irradiative and protected animals from liver intoxications. On the other hand, some anti-inflammative or anti-pyretic herbs such as Tripterygium wilfordii, Aconitum and Artemisiae species were proved to have immunosuppressive principles, some of them were now used clinically for the treatment of rheumatoid arthritis, chronic nephritis, systemic lupus erythematosis and various skin disorders. Pharmacological studies revealed that they have depressant effect on most of the humoral-immunity but not on the cell-mediated immunity. Some of them stimulated adrenal cortex functions and prolonged the survival time of transplanted allograft tissues.



[The effect of vitamin A and Astragalus on the splenic T lymphocyte-CFU of burned mice]

Pang SF
Chung Hua Cheng Hsing Shao Shang Wai Ko Tsa Chih (China) Jun 1989, 5 (2) p122-4, 159

In present study the effects of vitamin A and Astargalus on the splenic TL-CFU of mice were studied by means of T-lymphocytes colony formation in semi-solid culture in vitro and incorporation of 3H-TdR. Marked reduction of the responsive reaction of TL-CFU and T-lymphocyte transformation were found. The TL-CFU of the experimentally burned mice untreated with vitamin A (i.e. group 1) were significantly inhibited (p less than 0.005) in comparison with the unburned control group (i.e. group 4). And the TL-CFU of the experimentally burned mice treated with vitamin A (i.e. group 3) increased significantly (p less than 0.005) in comparison with group 1. Incorporation of 3H-TbR showed that vitamin A might accelerate the proliferation of the TL-CFU of the burned mice. It means that vitamin A might be regarded as an effective agent for the reversal of the inhibition of cell-mediated immunity in post-burned state, whether Ahstragalus plays a role in regulating immune inhibition needs further investigation.



Nutritional antioxidants and the modulation of inflammation: theory and practice.

Grimble RF
Institute of Human Nutrition, University of Southampton, UK.
New Horiz (United States) May 1994, 2 (2) p175-85

Highly potent substances are produced by the immune system. These substances include cytokines and oxidant molecules, such as hydrogen peroxide, free radicals, and hypochlorous acid. The purpose of immune cell products is to destroy invading organisms and damaged tissue, bringing about recovery. However, oxidants and cytokines can damage healthy tissue. Excessive or inappropriate production of these substances is associated with mortality and morbidity after infection and trauma, and in inflammatory diseases. Oxidants enhance interleukin-1, interleukin-8, and tumor necrosis factor production in response to inflammatory stimuli by activating the nuclear transcription factor, NF kappa B. Sophisticated antioxidant defenses directly and indirectly protect the host against the damaging influence of cytokines and oxidants. Indirect protection is afforded by antioxidants, which reduce activation of NF kappa B, thereby preventing up-regulation of cytokine production by oxidants. Cytokines increase both oxidant production and antioxidant defenses, thus minimizing damage to the host. While antioxidant defenses interact when a component is compromised, the nature and extent of the defenses are influenced by dietary intake of sulfur amino acids, for glutathione synthesis, and vitamins E and C. In animal studies, in vivo and in vitro responses to inflammatory stimuli are influenced by dietary intake of copper, zinc, selenium, N-acetylcysteine, cysteine, methionine, taurine, and vitamin E. Information from animal studies has yet to be fully translated into a clinical context. However, N-acetylcysteine, vitamin E, and a cocktail of antioxidant nutrients have reduced inflammatory symptoms in inflammatory joint disease, acute and chronic pancreatitis, and adult respiratory distress syndrome. Impaired antioxidant defenses may contribute to disease progression after infection with human immunodeficiency virus. Powerful arguments have been advanced for treatment with antioxidants to slow progression of acquired immunodeficiency syndrome. (76 Refs.)



Evaluation of zinc complexes on the replication of rhinovirus 2 in vitro.

Merluzzi VJ; Cipriano D; McNeil D; Fuchs V; Supeau C; Rosenthal AS; Skiles JW
Department of Immunology, Boehringer Ingelheim Pharmaceuticals Inc., Ridgefield, CT 06877.
Res Commun Chem Pathol Pharmacol (United States) Dec 1989, 66 (3) p425-40

The effect of zinc salts and complexes were evaluated on the replication of rhinovirus 2 in vitro. Zinc chloride inhibited the replication of rhinovirus 2 at concentrations between 3 and 12 micrograms/ml. Influenza virus was not affected. A number of zinc complexes were tested and compared to zinc chloride. The results indicated that the activity and toxicity of all zinc complexes in the rhinovirus cytopathogenic effect (CPE) assay were directly related to the amount of unbound zinc available.



Zinc gluconate and the common cold: a controlled clinical study.

Godfrey JC; Conant Sloane B; Smith DS; Turco JH; Mercer N; Godfrey NJ
Dartmouth College Health Service, Hanover, New Hampshire.
J Int Med Res (England) Jun 1992, 20 (3) p234-46

A report in 1984 on the success of zinc gluconate against common cold symptoms could not be confirmed in three subsequent studies, which are now known to have used formulations that inactivated zinc. A non-chelating formulation including glycine, which releases 93% of contained zinc into saliva, was tested in a randomized, placebo-controlled, double-blind trial in 73 young adults. Efficacy was recorded in symptom diaries using a symptom severity rating. Patients' symptoms first appeared 1.34 days prior to entry to the study in both groups. Disappearance of symptoms occurred after an additional 4.9 days for zinc-treated patients versus 6.1 days for placebo-treated patients. A difference was noted in the efficacy of treatment if it was started 1 day after symptom onset: cold duration was an additional 4.3 days in zinc-treated patients compared with 9.2 days for placebo-treated patients. Cough, nasal drainage and congestion were the symptoms most affected, and only mild side-effects were noted.



Prophylaxis and treatment of rhinovirus colds with zinc gluconate lozenges.

Al-Nakib W; Higgins PG; Barrow I; Batstone G; Tyrrell DA
MRC Common Cold Unit, Harvard Hospital, Salisbury, Wiltshire, U.K.
J Antimicrob Chemother (England) Dec 1987, 20 (6) p893-901

Following a tolerance study, double-blind placebo controlled trials were conducted to determine the prophylactic effect of zinc gluconate lozenges on rhinovirus challenge and, in a third study, their therapeutic efficacy when given at the start of colds caused by virus inoculation was tested. In the prophylaxis study a total of 57 volunteers received lozenges of either zinc gluconate (23 mg) (29 volunteers) or matched placebo (28 volunteers) every 2 h while awake during a period of four and a half days. They were challenged with 10(2) tissue culture infecting dose (TCID50) of human rhinovirus 2 (HRV-2) on the second day of medication, and were monitored daily for symptoms and signs of colds and laboratory evidence of infection. Zinc reduced the total mean clinical score from 8.2 in the placebo group to 5.7 and the reduction of the mean clinical score was statistically significant on the second day after virus challenge. In the therapeutic study 69 volunteers were inoculated with 10(2) TCID50 of HRV-2 and those who developed cold symptoms were randomly allocated to receive either zinc gluconate lozenges (six volunteers) or matched placebo lozenges (six volunteers) every two hours they were awake for six days. Treatment of colds with zinc reduced the mean daily clinical score and this was statistically significant on the fourth and fifth day of medication. Similarly, medication also reduced the mean daily nasal secretion weight and total tissue count and these reductions were statistically significant on days two and six for nasal secretion weights and days four to six of medication for tissue counts when compared with placebo.



Reduction in duration of common colds by zinc gluconate lozenges in a double-blind study.

Eby GA; Davis DR; Halcomb WW
Antimicrob Agents Chemother (United States) Jan 1984, 25 (1) p20-4

As a possible treatment for common colds, we tested zinc gluconate lozenges in a double-blind, placebo-controlled, clinical trial. One 23-mg zinc lozenge or matched placebo was dissolved in the mouth every 2 wakeful h after an initial double dose. After 7 days, 86% of 37 zinc-treated subjects were asymptomatic, compared with only 46% of 28 placebo-treated subjects (P = 0.0005). Side effects or complaints were usually minor and consisted mainly of objectionable taste and mouth irritation. Zinc lozenges shortened the average duration of common colds by about 7 days.



Antivirals for the chemoprophylaxis and treatment of influenza.

Van Voris LP; Newell PM
Division of Infectious Diseases, Hamot Medical Center, Erie, PA.
Semin Respir Infect (United States) Mar 1992, 7 (1) p61-70

Influenza virus infections are one of the leading causes of morbidity and mortality in the United States. Several antiviral agents, amantadine, rimantadine, and ribavirin, have been shown to be either therapeutically or prophylactically effective in influenza virus infections. Amantadine and rimantadine are effective, via the oral route, in treating and preventing influenza A infections. Aerosolized preparations of amantadine and rimantadine have also shown therapeutic efficacy against influenza A. Oral ribavirin has slight therapeutic efficacy in influenza A, but has also shown promising results in therapy of influenza B infections. Aerosolized ribavirin has also shown promise in treatment of patients who are severely ill with influenza A and B.



Utilization of pulse oximetry for the study of the inhibitory effects of antiviral agents on influenza virus in mice.

Sidwell RW; Huffman JH; Gilbert J; Moscon B; Pedersen G; Burger R; Warren RP
Institute for Antiviral Research, Utah State University, Logan 84322-5600.
Antimicrob Agents Chemother (United States) Feb 1992, 36 (2) p473-6

Pulmonary disease in mice induced by influenza virus was monitored by measurement of oxygen saturation (SaO2) in blood with a pulse oximeter. The SaO2 declined in inverse proportion to the viral inoculum. The known antiviral agent ribavirin inhibited the SaO2 decline, prevented death, lowered lung consolidation, and reduced the level of recoverable virus. Pulse oximetry is an effective means of monitoring murine influenzal disease and can be used in the study of potential antiviral drugs.



Further studies with short duration ribavirin aerosol for the treatment of influenza virus infection in mice and respiratory syncytial virus infection in cotton rats.

Gilbert BE; Wyde PR; Ambrose MW; Wilson SZ; Knight V
Department of Microbiology and Immunology, Baylor College of Medicine, Houston, TX 77030.
Antiviral Res (Netherlands) Jan 1992, 17 (1) p33-42

Ribavirin aerosol administration has been shown to be effective in the treatment of respiratory syncytial virus (RSV) infections in infants and in influenza A and B virus infections in young adults. Long treatment schedules and potential for environmental contamination have stimulated the search for alternative dosing schedules. Thus, we attempted to determine the length of time of ribavirin aerosol necessary for effective treatment of influenza and RSV. In RSV-infected cotton rats, aerosolization for just 30 min with high-dose ribavirin (HDR:60 mg ribavirin/ml in reservoir), 3 times daily, reduced viral lung titers/gm of tissue by 1.1 log10. In influenza virus-infected mice, 15 min of aerosolized HDR, 3 times daily, was effective in reducing both mortality and pulmonary virus titers (1.1 log10 reduction). When the intervals between aerosol administration each day were equally divided (i.e., q.8 h), the treatments were most effective. Treatment for 45 min, once daily, was not as effective as divided doses. Calculations of ribavirin concentrations in respiratory secretions following 15 min treatment in mice with HDR indicated that drug levels dropped below the ED50 for influenza viruses after about 9 h. A daily dosage of ribavirin, estimated to be 8-15 mg/kg, was effective for the treatment of influenza and RSV infections.



High dose-short duration ribavirin aerosol treatment--a review.

Knight V, Gilbert BE, Wyde PR, Englund JA
Center for Biotechnology, Baylor College of Medicine, Houston, Texas 77381.
Bull Int Union Tuberc Lung Dis 1991 Jun-Sep;66(2-3):97-101

A high-dose, short-duration treatment with ribavirin aerosol consisting of a three-fold increase in concentration of drug (60 mg versus 20 mg of ribavirin per mL in the liquid reservoir of the generator administered for about one-third the time of the standard treatment) was as effective as the standard dosage in the treatment of experimental influenza A and B infections in mice and in the treatment of experimental respiratory syncytial virus infection in cotton rats. Despite some minor pulmonary intolerance, it was considered to be suitable for use in treatment of patients with severe chronic pulmonary disease, and it was well-tolerated and apparently effective in the treatment (by face mask and endotracheal tube) of infants with bronchiolitis principally caused by respiratory syncytial virus infection. Pharmacokinetic studies in mice revealed very high concentrations of drug in the lungs, about triple the level with the standard dose, with similar blood and brain concentrations. Ribavirin concentrations were similarly high in respiratory secretions of infants given the triple dose.



Viral pneumonia.

Greenberg SB
Department of Medicine, Baylor College of Medicine, Houston, Texas.
Infect Dis Clin North Am 1991 Sep;5(3):603-21

Viral pneumonias are common in infants and young children but rare in adults. Respiratory syncytial virus (RSV) and para-influenza viruses are the most frequent viral pathogens in infants and children. Influenza virus types A and B account for over one half of viral pneumonias in adults. Immunocompromised hosts are susceptible to pneumonias caused by cytomegalovirus (CMV) and other herpesviruses, as well as rubeola and adenovirus. Diagnosis of viral pneumonia depends on appropriate viral cultures and acute and convalescent sera for specific antibodies. Superinfection with bacteria is common in adults. Anti-viral therapy is available for several respiratory viruses. Ribavirin, amantadine/rimantadine, interferon alpha, and acyclovir are antiviral drugs that may be of benefit in treatment and prophylaxis. Prevention of viral pneumonia will depend upon improved viral immunization practices.



Aerosol and intraperitoneal administration of ribavirin and ribavirin triacetate: pharmacokinetics and protection of mice against intracerebral infection with influenza A/WSN virus.

Gilbert BE; Wyde PR; Wilson SZ; Robins RK
Department of Microbiology and Immunology, Baylor College of Medicine, Houston, Texas 77030.
Antimicrob Agents Chemother (United States) Jul 1991, 35 (7) p1448-53

Ribavirin is active in vitro but not in vivo against a number of viruses capable of causing encephalitis. Ribavirin triacetate (RTA), a lipophilic derivative, has been reported to be more effective than ribavirin in protecting animals from encephalitis. By using an influenza A/WSN virus encephalitis model, we demonstrated that RTA administered by small-particle aerosol was able to decrease the death rate and increase the time of survival. To determine if this beneficial effect was due to increased delivery of drug, the pharmacokinetic properties of ribavirin and RTA when administered as an aerosol or by intraperitoneal injection were examined. Aerosol administration of ribavirin or RTA gave significantly higher concentrations of ribavirin in the lungs and serum of mice than did intraperitoneal injection. There was no difference, however, in ribavirin levels when either ribavirin or RTA was administered by small-particle aerosol. In brain tissue, ribavirin concentrations increased with time and did not appear to decrease as rapidly as in lungs and serum. Mean peak ribavirin concentrations in the brain were higher following aerosol administration of ribavirin than RTA, and both were higher than that following intraperitoneal injection of either drug. Administration of ribavirin or RTA by intraperitoneal injection failed to protect mice from a lethal intracerebral inoculation of influenza A/WSN virus, while aerosolized RTA did protect mice. The pharmacokinetics of ribavirin in brain tissue following aerosol administration of either drug did not explain the advantage of RTA over ribavirin in protecting mice from intracerebral infection with influenza A/WSN virus.



Antiviral drug therapy.

Goodpasture HC
University of Kansas School of Medicine-Wichita.
Am Fam Physician (United States) Jan 1991, 43 (1) p197-204

Major advances in molecular virology have led to the development of new antiviral compounds. These drugs include ribavirin, used in the treatment of severe respiratory syncytial virus infection in children; amantadine, used in the prophylaxis and treatment of influenza A infection; acyclovir, used in a variety of herpesvirus infections, including primary gingivostomatitis, genital herpes and herpes zoster; ganciclovir, used in the treatment of retinitis due to cytomegalovirus, and zidovudine, used in the prophylaxis and treatment of human immunodeficiency virus infection.



Molecular mechanisms of action of ribavirin.

Patterson JL; Fernandez-Larsson R
Division of Infectious Diseases, Children's Hospital, Boston, Massachusetts 02115.
Rev Infect Dis 1990 Nov-Dec;12(6):1139-46

Ribavirin (1-beta-D-ribofuranosyl-1,2,4-triazole-3-carboxamide) is a broad-spectrum antiviral agent whose molecular mode of action remains remarkably controversial. This antiviral agent was approved by the U.S. Food and Drug Administration in 1986 for use as an aerosol for infants with serious infections due to respiratory syncytial virus. Ribavirin is and has been under clinical investigation for activity against a variety of viral illnesses, including those due to influenza virus, Lassa fever virus, Hantaan virus, and human immunodeficiency virus (HIV). There has been a great deal of clinical interest in the utilization of ribavirin for treatment of infections due to HIV. It has been reported to slow the development of AIDS in HIV-infected patients. We describe here the major mechanisms of action of this newly licensed antiviral agent.



New acquisitions in the chemotherapy of viral infections.

De Clercq E
Department of Human Biology, Rega Institute for Medical Research, Katholieke Universiteit Leuven, Belgium.
Verh K Acad Geneeskd Belg 1990;52(1):69-99

The development of new antiviral agents has gained increasing momentum. It has kept pace with the identification of specific sites ("targets") in the virus replicative cycle at which potential antiviral drug can interact. The current armamentarium of available antiviral drugs consists of amantadine and rimantadine (against influenza A), ribavirin (against respiratory syncytial virus infection), idoxuridine and trifluridine (against herpetic keratitis), vidarabine and acyclovir (against herpes simplex virus infections), ganciclovir (against cytomegalovirus infections) and Retrovir (against AIDS). Various new compounds have been found which selectively inhibit those viruses [i.e. adenovirus, varicella-zoster virus, thymidine kinase-deficient (TK-) herpes simplex virus strains, and rhinoviruses] that are insensitive or poorly sensitive to the presently available antivirals. Several new compounds have also proven active against human immunodeficiency virus, the causative agent of AIDS; and, as a spin-off of the search for anti-AIDS drugs, new agents may also be expected that are effective against other retrovirus infections as well as hepadnavirus (i.e. hepatitis B virus) infections. (86 Refs.)



Comparison of oral and aerosol ribavirin regimens in the high risk elderly

Bernstein JM; Liss H; Erk SD
Department of Medicine, Wright State University School of Medicine, Dayton, OH.
J Clin Pharmacol 1989 Dec;29(12):1128-34

A comparison of different regiments of ribavirin (R), administered either orally or by aerosol, was performed in 16 elderly subjects (13 men, 3 women, mean age 63 +/- 8 years) considered to be in the "high-risk" category for complications from influenza as defined by the Centers for Disease Control. The subjects were divided into four groups. Group O-600 received 600 mg orally R every 8 hours for 48 hours followed by 200 mg every 8 hours for 72 hours for a total dose of 5.4 g (22.1 mmol). Group O-800 received 800 mg oral R every 8 hours for 24 hours followed by 400 mg every 12 hours for 96 hours for a total dose of 4.1 g (22.9 mMoles). Group A-40 received R (40 mg/ml) aerosolized through a small particle aerosol generator for 6 hours every 12 hours for 96 hours, yielding an average delivered dose of 6.2 g (25.4 mMoles) R. Group A-60 received aerosolized R (60 mg/mL) for 2 hours every 8 hours for 96 hours, yielding an average delivered dose of 4.6 g (18.8 mMoles) R. No hematologic or other laboratory abnormalities were associated with any of the regimens. Group O-800 and O-600 reached mean peak plasma R levels of 11.8 microM and 5.3 microM, respectively, after 18 hours of therapy. Subsequent administration of 20 mg R every 8 hours was sufficient to maintain a plasma R level greater than 7 microM. Among the aerosol groups, group A-40 approached steady state plasma R levels (8-10 microM) more quickly than group A-60.



Comparative activities of several nucleoside analogs against influenza A, B, and C viruses in vitro.

Shigeta S; Konno K; Yokota T; Nakamura K; De Clercq E
Department of Bacteriology, Fukushima Medical College, Japan.
Antimicrob Agents Chemother. 1988 Jun;32(6):906-11.

A set of 20 nucleoside analogs were examined for their inhibitory effects on the cytopathogenicity and growth of influenza virus type A, B, and C strains in Madin-Darby canine kidney (MDCK) cells. Among the compounds evaluated, pyrazofurin, 3-deazaguanine, ribavirin, carbodine, and cyclopentenyl cytosine inhibited viral cytopathogenicity at concentrations that were lower than those found cytotoxic for the MDCK cells. No differences were observed in the 50% effective doses (based on inhibition of viral cytopathogenicity) of these five compounds for a number of influenza virus type A (subtypes H1N1 and H3N2), B, and C strains. Pyrazofurin showed the lowest 50% effective dose (0.15 microgram/ml), which was about 20- to 30-fold lower than those of the other four compounds. The selectivity indices of the five compounds, calculated as the ratio of the 50% cytotoxic dose (determined by trypan blue exclusion) to the 50% effective dose, were greater than 100. When the selectivity indices were calculated as the ratios of the 50% inhibitory doses for cellular RNA synthesis to the 50% effective doses, they were greater than 100 for ribavirin, pyrazofurin, and 3-deazaguanine but less than 2 for carbodine and cyclopentenyl cytosine. All five compounds inhibited the growth of influenza virus types A and B in MDCK cells at a concentration which was well below their cytotoxicity threshold for MDCK cells and, therefore, deserve further exploration for their potential in the treatment of influenza virus type A, B, and C infections.



Antiviral drugs for common respiratory diseases. What's here, what's to come.

Johnson DC
Department of Pediatrics, Michael Reese Hospital, Chicago, IL 60616.
Postgrad Med (United States) Feb 1 1988, 83 (2) p136-9, 142-3, 146-8

Progress is being made in the development of drugs for the prevention and treatment of viral respiratory infections. Two drugs currently available to clinicians are amantadine (Symmetral) and ribavirin (Virazole). Oral amantadine is effective for both treatment and prevention of uncomplicated influenza A infections. Although vaccination continues as the mainstay of influenza prevention, amantadine is useful for unvaccinated patients if complications are likely. When used for treatment, it must be started within the first 48 hours of illness. Ribavirin appears to be safe for treatment of respiratory syncytial virus infections in nonintubated infants. It must be delivered by aerosol in a hospital setting. Patients at risk for complications should be given the drug as early as possible in the course of the disease. Efficacy has yet to be proven in intubated patients, but the drug is probably safe to use with proper supervision. On the horizon are rimantadine and the interferons. Rimantadine is similar to amantadine in its action and indications for use and has a lower incidence of side effects. The interferons have not been the hoped-for panacea for viral respiratory infections but may be useful in a nasal spray for the prevention of colds caused by rhinovirus.



Oral ribavirin treatment of influenza A and B.

Stein DS; Creticos CM; Jackson GG; Bernstein JM; Hayden FG; Schiff GM; Bernstein DI
Antimicrob Agents Chemother. 1987 Aug;31(8):1285-7.

A loading dose and short-term administration of oral ribavirin significantly improved symptoms and signs of influenza type A or B infection in 25 patients. The antiviral effect was not significant. No adverse clinical effects or significant laboratory values were observed. Oral treatment of patients with influenza A or B infection might be possible with ribavirin.



Clinical review of ribavirin.

Eggleston M
Infect Control (United States) May 1987, 8 (5) p215-8

The recent approval of ribavirin aerosol for the treatment of severe respiratory syncytial virus (RSV) in infants and young children is a significant addition to the antiviral drugs available today. When administered as an aerosolized form by face mask or mist tent for 20 to 21 hours per day, ribavirin effectively decreases the symptoms of RSV infection and the shedding of RSV virus. Studies of other viral infections such as viral hepatitis, influenza A and B, Lassa fever, genital herpes, and herpes zoster have demonstrated promising, but inconclusive results. Further studies are needed to justify ribavirin therapy for these indications.



Clinical use of antiviral drugs.

Nahata MC
Drug Intell Clin Pharm 1987 May;21(5):399-405

Remarkable progress has been made in antiviral chemotherapy. Six approved antiviral drugs are now available for the treatment of various viral infections. Trifluridine, idoxuridine and vidarabine are all effective in patients with herpes keratitis; trifluridine is preferred due to its low toxicity. Acyclovir is the drug of choice in patients with infections due to herpes simplex viruses, including genital herpes, herpes encephalitis, and neonatal herpes, and infections due to varicella-zoster virus. Amantadine is the only drug currently available for prophylaxis and treatment of influenza A, but an investigational drug, rimantadine, appears to be equally effective and less toxic than amantadine. Ribavirin is the most recently approved antiviral agent for the treatment of respiratory syncytial virus infections. Numerous antiviral drugs are being studied in patients with acquired immunodeficiency syndrome. Although currently available drugs have improved our ability to manage a variety of viral illnesses, much needs to be learned about specific dosage guidelines based on the studies of pharmacokinetics, pharmacodynamics, potential adverse effects and viral resistance, and the role of combination therapy to optimize therapy.



Protection of mice from lethal influenza virus infection with high dose-short duration ribavirin aerosol.

Wyde PR; Wilson SZ; Gilbert BE; Smith RH
Antimicrob Agents Chemother (United States) Dec 1986, 30 (6) p942-4

An aerosol generated from a reservoir containing 60 mg of ribavirin per ml given for 2 h twice daily for 4 days afforded the same high level of protection against lethal influenza virus infection of mice as a longer, conventional treatment schedule (20 mg/ml given for 11 h daily for 4 days). Incremental decreases in ribavirin concentration made while maintaining the 2-h intermittent schedule provided progressively less protection of mice. Mice exposed to the 60-mg/ml doses had significantly increased pulmonary and serum drug levels when compared with mice given 20 mg of drug per ml, these increases were transient, and no evidence of pulmonary intolerance was detected. These studies suggest that protective effects of ribavirin against influenza virus infection can be achieved without untoward effects if higher doses and shorter periods of administration are used.



Ribavirin: a clinical overview.

Fernandez H; Banks G; Smith R
Eur J Epidemiol. 1986 Mar;2(1):1-14

Ribavirin, a broad spectrum, non-interferon-inducing virustatic chemotherapeutic agent, demonstrates activity against a wide range of RNA and DNA viruses, including the retrovirus known to cause the acquired immune deficiency syndrome. The drug's proposed mechanism of action, as well as pharmacokinetics are discussed, and preclinical toxicity, safety and clinical efficacy studies are presented. To date, the best success has occurred in the use of ribavirin to treat respiratory syncytial virus infection in infants and young children and to treat influenza A and B virus infections in young adults. Viral infections, particularly viral pneumonia, are often life-threatening in infants with severe combined immunodeficiency disease (SCID), and ribavirin aerosol has been used successfully to treat respiratory syncytial virus and parainfluenza virus infection of immunodeficient children. Special note is taken of ribavirin's clinical benefit in treating severe and life-threatening infections caused by the Lassa fever virus and the significant improvement over either the use of immune plasma or supportive therapy alone. Indeed, ribavirin thus emerges as the first antiviral drug that is able to reduce mortality in a highly lethal systemic disease by more than 90%. Additional studies demonstrate the drug's efficacy in acute viral hepatitis, herpesvirus infections, and measles. Controlled clinical trials are underway to test the drug in patients infected with the AIDS virus.



Effect of ribavirin triphosphate on primer generation and elongation during influenza virus transcription in vitro.

Wray SK; Gilbert BE; Knight V
Antiviral Res (Netherlands) Feb 1985, 5 (1) p39-48

These studies examine the effect of ribavirin triphosphate (RTP) on two replicative functions associated with influenza virus nucleocapsids, primer generation and its subsequent elongation. To study primer generation influenza virus cores were added to beta-globin mRNA in the presence of only [32P]GTP. To examine elongation, ATP and CTP were added to the reaction mixture to permit limited elongation, and products from both reactions were separated on polyacrylamide gels and quantified. Under these conditions, the 50% inhibitory concentration of RTP for primer generation was 3.0 mM, and the 50% inhibitory concentration for elongation was 0.6 mM. RNA polymerase activity associated with cores isolated from clinical strains of influenza A and B viruses reacted as did the laboratory strain of influenza virus and was equally susceptible to inhibition by RTP.



Ribavirin

Conner CS
Drug Intell Clin Pharm 1984 Feb;18(2):137-8

Despite the plethora of antibiotics available for the treatment of bacterial infections, very few agents have been developed to treat viral diseases. Ribavirin (Virazole) is a triazole nucleoside antiviral agent that produces selective antiviral effects against a broad spectrum of RNA and DNA viruses. The drug has been effective in the treatment of naturally occurring influenza A and B infections when administered by aerosol; oral administration has been ineffective. Ribavirin aerosol therapy also has proven effective to reduce symptoms of respiratory syncytial virus infections in young adults and hospitalized neonates. Ribavirin aerosol may be the first antiviral agent to treat these common diseases.



[Immunomodulating activity of ethanol-water extracts of the roots of Echinacea gloriosa L., Echinacea angustifolia DC. and Rudbeckia speciosa Wenderoth tested on the immune system in C57BL6 inbred mice]

Bukovsky M; Vaverkova S; Kostalova D; Magnusova R
Katedra biochemie a mikrobiologie Farmaceutickej fakulty Univerzity Komenskeho, Bratislava.
Cesk Farm (Czech Republic) Aug 1993, 42 (4) p184-7

The ethanolic extract from the roots Echinacea gloriosa L. (Moench), Echinacea angustifolia DC. and Rudbeckia speciosa Wenderoth shows immunomodulating activity. It was seen on the seventh day after five days of in vivo treatment of mice. The most marked immunostimulatory effect was observed on the lysosomal and peroxidal activity of peritoneal macrophages, and splenic cells after in vivo treatment with the ethanolic xtract of the roots of R. speciosa Wenderoth.



Application of purified polysaccharides from cell cultures of the plant Echinacea purpurea to mice mediates protection against systemic infections with Listeria monocytogenes and Candida albicans.

Roesler J, Steinmuller C, Kiderlen A, Emmendorffer A, Wagner H, Lohmann-Matthes ML
Fraunhofer-Institut, Department of Immunobiology, Hannover, F.R.G.
Int J Immunopharmacol. 1991;13(1):27-37.

Purified polysaccharides from cell cultures of the plant Echinacea purpurea were investigated for their ability to enhance phagocytes' activities regarding nonspecific immunity in vitro and in vivo. Macrophages (M phi) from different organ origin could be activated to produce IL-1, TNF alpha and IL-6, to produce elevated amounts of reactive oxygen intermediates and to inhibit growth of Candida albicans in vitro. Furthermore, in vivo the substances could induce increased proliferation of phagocytes in spleen and bone marrow and migration of granulocytes to the peripheral blood. These effects indeed resulted in excellent protection of mice against the consequences of lethal infections with one predominantly M phi dependent and one predominantly granulocyte dependent pathogen, Listeria monocytogenes and C. albicans, respectively. Specific immune responses to sheep red blood cells (antibody production) and to listeria (DTH) were not affected by the polysaccharides. The possibility of clinical use is discussed.



Macrophage activation by the polysaccharide arabinogalactan isolated from plant cell cultures of Echinacea purpurea.

Luettig B; Steinmuller C; Gifford GE; Wagner H; Lohmann-Matthes ML
Fraunhofer Institute fur Toxikologie, Abt. Immunbiologie, Hannover, Federal Republic of Germany.
J Natl Cancer Inst (United States) May 3 1989, 81 (9) p669-75

In this study, acidic arabinogalactan, a highly purified polysaccharide from plant cell cultures of Echinacea purpurea, with a molecular weight of 75,000, was effective in activating macrophages to cytotoxicity against tumor cells and micro-organisms (Leishmania enriettii). Furthermore, this polysaccharide induced macrophages to produce tumor necrosis factor (TNF-alpha), interleukin-1 (IL-1), and interferon-beta 2. Arabinogalactan did not activate B cells and did not induce T cells to produce interleukin-2, interferon-beta 2, or interferon-gamma, but it did induce a slight increase in T-cell proliferation. When injected ip, this agent stimulated macrophages, a finding that may have therapeutic implications in the defense against tumors and infectious diseases.



Macrophage activation and induction of macrophage cytotoxicity by purified polysaccharide fractions from the plant Echinacea purpurea.

Stimpel M; Proksch A; Wagner H; Lohmann-Matthes ML
Infect Immun. 1984 Dec;46(3):845-9.

Purified polysaccharides (EPS) prepared from the plant Echinacea purpurea are shown to strongly activate macrophages. Macrophages activated with these substances develop pronounced extracellular cytotoxicity against tumor targets. The activation is brought about by EPS alone and is independent of any cooperative effect with lymphocytes. Also the production and secretion of oxygen radicals and interleukin 1 by macrophages is increased after activation with EPS. Cells of the macrophages lineage seem to be the main target for the action of these polysaccharides. EPS has no effect on T lymphocytes. B lymphocytes show a comparatively modest proliferation after incubation with E. purpurea EPS. Thus, these compounds, which are at least in tissue culture completely nontoxic, may be suited to activate in vivo cells of the macrophage system to cytotoxicity. They may therefore be of relevance in tumor and infectious systems.



Combined antiviral and antimediator treatment of rhinovirus colds.

Gwaltney JM Jr
Department of Internal Medicine, University of Virginia Health Sciences Center, Charlottesville 22908.
J Infect Dis 1992 Oct;166(4):776-82

An antiviral agent and two antiinflammatory compounds were used in a blinded, placebo-controlled study to treat experimental rhinovirus colds. Intranasal interferon-alpha 2b and ipratropium and oral naproxen were begun 24 h after rhinovirus inoculation. Treatment was continued three times a day for 4 days. Viral shedding (mean +/- SE) was 4.4 +/- 0.3 days for controls and 2.9 +/- 0.3 days for treated volunteers (P less than .003). Geometric mean virus titers were reduced in the treated group on all days (P = .02-.06). Serum antibody responses and postinfection geometric mean antibody titers were similar in both groups (P greater than .1). Colds developed in 6 of 16 treated and 7 of 8 control subjects (P = .05). Mean total symptom scores (P = .055), rhinorrhea (P less than .01), cough (P less than .01), and malaise (P less than .001) were reduced in treated subjects. Trends in reduction of nasal obstruction and sore throat also favored the treated group. Nasal secretion weights were 12.9 +/- 4.8 g in treated and 20.3 +/- 5.4 g in control subjects (P = .4). Medications were was tolerated.



[Common cold: diagnostic steps? Antibiotics?]

Auckenthaler R
Division des maladies infectieuses, Hopital cantonal universitaire, Geneve.
Ther Umsch (Switzerland) Apr 1992, 49 (4) p211-5

The common cold is caused by more than 100 virus types. However, the clinical manifestation is always similar with rhinorrhea, stuffiness, sneezing, pharyngitis, laryngitis and cough. The local inflammatory reactions are not due to the presence of virus but caused by locally produced inflammatory mediators. Bacterial superinfections may cause otitis or sinusitis. Bacterial nasopharyngitis has been described in children. This entity possibly exists also in adults. Traditional viral cultures are rarely positive and are not recommended in the daily routine. In children, antigen detection for adenovirus, respiratory syncytial virus, parainfluenza and influenza virus are recommended to confirm the viral etiology or for epidemiological surveillance. The presence of group-A streptococci must be proven by culture or antigen detection before treatment with penicillin. Antiviral treatment is limited to interferon or ribavirin. New antiviral substances are in development. Today, treatment of common cold is limited to symptomatic measures, and antibiotic treatment is not justified.



Alpha 2-interferon for the common cold.

Enlow ML, Haley CJ
Ann Pharmacother 1992 Mar;26(3):345-7

No abstract.



Managing viral upper respiratory infections.

Del Mar C
Aust Fam Physician 1991 May;20(5):557-61

The epidemiology of the common cold is reviewed with the aim of providing helpful advice for patients. Future management will include limiting the spread of the cold virus by attention to the mode of transmission and the development of anti-viral drugs, of which interferon holds the most promise.



Immunological barriers in the nose and paranasal sinuses.

Mygind N, Winther B
Acta Otolaryngol (Stockh) 1987 May-Jun;103(5-6):363-8

This review deals mainly with lymphocyte subsets in the human nasal mucosa, and with the common cold. Lymphocytes have recently been characterized in biopsy specimens by an immuno-histochemical method (the avidin-biotin, monoclonal antibody peroxidase technique). In summary, the overall T:B cell ratio was 3:1 and that of T helper cells to T suppressor was 2.5:1; topographical differences within the nasal mucosa were identified. Non-specific defence systems, such as interferon, provide some protection against rhinovirus infection, but most important is the presence of specific antibodies against a given antigenic type of virus. Recent results have suggested that a rhinovirus infection does not cause a marked destruction of the epithelial lining, that it is spotty in the nasal mucosa, and that it is most prominent in the nasopharynx. Increased knowledge about the site of infection and how symptoms are produced is essential for a rational approach to the development of anti-viral therapy.



Interferon for the treatment of infections.

Ho M
Annu Rev Med (United States) 1987, 38 p51-9

Interferon, both natural and recombinant, has been shown in controlled clinical studies to be effective against herpes simplex virus infections, herpes zoster, the common cold caused by rhinoviruses, and some papilloma virus infections. In some cases, it is in competition with other antivirals, and in others its precise clinical indication is still unclear. Thus, further work and developments are required before interferon becomes a clinically recognized antiviral agent.



Effect of Astragalus membranaceus on electrophysiological activities of acute experimental coxsackie B-3 viral myocarditis in mice

Rui T; Yang YZ; Zhou TS
Shanghai Institute of Cardiovascular Disease.
Chung Kuo Chung Hsi I Chieh Ho Tsa Chih (China) May 1994, 14 (5) p292-4, 262

A murine model for observing the effect of Astragalus membranaceus (AM) on electrophysiological activity of the right ventricular myocardium was developed in 4 week-old male BALB/c mice infected with Coxsackie B3 virus (CB3V). The conventional microelectrode technique and real-time microcomputer data processor system was used. The survival rate in infected-AM treated mice was significantly higher and the percentage of abnormal action potential was much lower than those in control mice (P < 0.05 and < 0.01 respectively). Some abnormal electrophysiological parameters, such as APA, OS and Vmax in infected myocardium were found to be improved by AM treatment. Single dose of AM did not show beneficial effect in murine myocardium infected with CB3V. The results suggested that AM might be valuable in the prevention and treatment of acute myocarditis involving Coxsackie B3 virus.



Efficacy and safety of the standardized ginseng extract G 115 for potentiating vaccination against common cold and/or influenza syndrome

Scaglione F, Cattaneo G, Alessandria M, Cogo R
Department of Pharmacology, University of Milan, Italy.
Drugs Exp Clin Res 1996;22(2):65-72
[Corrected] [published erratum appears in Drugs Exp Clin Res 1996;22(6):338]

The aim of the study was to determine the properties of a standardized extract of ginseng root in inducing a higher immune response in vaccination against influenza. Attention was also paid to the common cold in this multicentre, two-arm, randomized, placebo-controlled, double-blind investigation. A total of 227 volunteers who visited 3 private practices in Milan received daily oral capsule doses of either placebo (113) or 100 mg of standardized ginseng extract Ginsana G115 (114) for a period of 12 weeks within which they received an anti-influenza polyvalent vaccination at week 4. As a result, while the frequency of influenza or common cold between weeks 4 and 12 was 42 cases in the placebo group, it was only 15 cases in the G115 group, the difference being statistically highly significant (p < 0.001). Whereas antibody titres by week 8 rose to an average of 171 units in the placebo group, they rose to an average of 272 units in the G115 group (p < 0.0001). Natural killer (NK) activity levels at weeks 8 and 12 were nearly twice as high in the G115 group as compared to the placebo group (p < 0.0001). In all the volunteers, laboratory values of 24 safety parameters showed no significant differences between the end and the beginning of the 12-week study in either of the groups. There were only 9 adverse events in the study, the principal one being insomnia.



An emerging green pharmacy: Modern plant medicines and health

Laboratory Medicine (USA), 1996, 27/3 (170-176)

Recently plants have reemerged as sources of new pharmaceuticals. Drugs derived from plants are used to treat conditions ranging from arthritis and malaria to leukemia and ovarian cancer. Some of today's treatments use herbs directly. Researchers also are studying a variety of foods for their potential medicinal benefits. More and more consumers are buying herbal medications in the form of food supplements to use as analgesics, sedatives, or immune system stimulants. Although a few plants may cause serious adverse reactions, many herbal preparations are considered to be safe and effective in moderation. This is the third article in a four-part continuing education update series on botany. Other articles focus on the use of plants to clean up the environment, the historical use of plant therapies, and poisonous plants. Following this series, participants should be able to identify plants used medicinally today and throughout history. They will recognize the role of plants in the environment and be able to identify toxic plants in the laboratory.



Immunity in myocardiac hypertrophy rat and effect of total saponins of panax ginseng in vivo and in vitro

Chinese Pharmacological Bulletin (China), 1996, 12/1 (84-86)

The model of rat myocardiac hypertrophy through stricture on abdominal aorta partly by operation showed that proliferation of T cell in thymus and spleen decreased and IL-2 secretion reduced markedly when rat blood pressure increased and the wall of left ventricular thickened. Total saponins of panax ginseng (TSPG 50 mg.kg-1.d-1, sc ) could harmonize the higher blood pressure and increase the level of immunity, suggesting TSPG may be used to strengthen the heart function as well as immunity.



Treatment of experimental coxsackie B-3 viral myocarditis with astragalus membranaceus in mice

Yang YZ, Jin PY, Guo Q, Wu WZ, Pu SY, Chen HZ, Yang JH, Wang KQ, Shi JY, Gong ZX, et al
Shanghai Institute of Cardiovascular Disease, Zhongshan Hospital, Shanghai Medical University.
Chin Med J (Engl) 1990 Jan;103(1):14-8

A murine model system for observing the effect of Astragalus Membranaceus (AM) on experimental myocarditis caused by Coxsackie B-3 virus (CB3V) was developed in 4-week-old male BALB / C mice. Gross, histopathologic and ultrastructural examinations of the infected-AM treated group showed that the severity and involved area of the myocardial lesions became milder and smaller than those in the infected-NS treated mice. The total lesion area, and the total lesion area / total myocardial area examined (%) and virus titer in the former group were also smaller and lower than those in the latter group. The results suggest that AM is effective in the inhibition of Coxsackie B virus propagation and protection of myocardium in mouse myocarditis.



Effect of Astragalus membranaceus injecta on coxsackie b-2 virusinfected rat beating heart cell culture

Yang YZ; Guo Q; Jin PY; Pu SY; Chen HZ; Cheng JR; Jin YX; Gong ZX; Shen JY
Chin. Med. J. (Peking) (China), 1987, 100/7 (595-602)

Astragalus membranaceus (AM) injecta protects rat beating heart cells experimentally infected with Coxsackie B-2 virus as evaluated for changes in release of cardiac enzymes (lactate dehydrogenase and aspartate aminotransferase). Heart beat rate, cytopathic effects, cardiac cellular damage as measured by cytotoxicity assay, virus titer, and ultrastructure were monitored. Significant protective effects were demonstrated when AM was given 1-9 hours post-infection. The results suggest that AM may be valuable in prophylaxis and treatment of acute Coxsackie virus caused myocarditis



Sambucol(tm) inhibited several straing of influenza virus and reduced symptoms during an outbreak of Influenza B Panama

Weizmann Institute of Science 2-15-94

Sambucol, a new product based on the fruit of the black elder, inhibited the replication of influenza virus types A and B: A/Beijing 32/92 (H3N2), A/Singapore 6/86 HlN1), B/Panama 45/90, B/Yamagata 16/88 and B/Ann Arbor 1/86 in Madin-Darby canine kidney cells (MDCK). A placebo-controlled, double blind study was conducted on a group of individuals living in a kibbutz during an outbreak of influenza B/Panama 45/90 characterized by hemagglutination tese. Patients who were admitted to the study had at least three of the following symptoms of less than 24 h duration: fever > 38 C, myalgia, nasal discharge and cough. Fever, feeling of improvement and complete cure were recorded during 6-days. Sera obtained in the acute and convalescent phases were tested for the presence of antibodies to influenza A and B, respiratory syncytia! and adeno viruses. Convalescent phase serologies showed higher mean and mean geometric hemagglutination inhibirion titers eo influenza B in the Sambucol group than in the control group, in spite of the more rapid recovery. A complete cure was achieved within 2 toe 3 days in nearly 90% of the Sambucol group whereas recovery took at least 6 days in the placebo group (p <0.001). In the absence of any medication against influenza B virus and considering its low cost and absence of side-effects, Sambucol may offer the possibility for safe treatment for influenza.



The effect of Sambucol(tm) on HIV infection in vitro

Congress of Microbiology 2-6-95

Sambucol, a new product based on the fruit of the black elder, contains a high amount of three flavonoids. Sambucol exhibited antiviral activity against various strains of influenza virus (both A and B), herpes virus type 1 and parainfluenza viruses. In this study we tested the ability of Sambucol to inhibit the infection of laboratory HIV strains as well as clinical HIV isolates in CD4+ cell lines (CEM and Molt 4) and human peripheral blood lymphocytes. For this purpose HIV was pre-incubated with two dilutions of Sambucol before being added to the cells. We determined a significant reduction in the infectivity of HIV strains (ELI, LAI, HIV IIIb) in the presence of Sambucol, by measuring the level of HIV core antigen p24 in supernatants of the infected cultures, as compared with controls without Sambucol. We did not detect HIV-antigen 5 and 9 days post infection in cultures infected with patient isolates which were previously treated with Sambucol. Such an approach may have a practical application in designing a simple or combined viral intervention therapy for individuals already exposed to the virus.




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